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Browsing by Author "Hadiyal, S. D."

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Design and rapid microwave irradiated one-pot synthesis of tetrahydropyrimidine derivatives and their screening in vitro antidiabetic activity

Lalpara, J. N.; Hadiyal, S. D.; Radia, A. J.; Dhalani, J. M.; Dubal, G. G. (Taylor & Francis Group, LLC / Polycyclic Aromatic Compounds, 2020-12-01)

A rapid and efficient method has been developed for one-pot synthesis of some newly designed tetrahydropyrimidine derivatives with aid of 1,3,4-oxadiazole containing aldehyde, substituted acetoacetanilide and thiourea/guanidine ...
Growth and Characterization of Dicoumarole Derivative

Parmar, S. K.; Gohil, H. K.; Vyas, P. M.; Hadiyal, S. D.; Patel, A. H. (International Journal of Advance and Innovative Research, 2018)

The Dicoumarole derivative 4-amino-3-((4-amino-2-oxo-2H-chromen-3-yl)(3-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl)methyl)-2H-chromen-2-one obtain by crystal growth by slow evaporation solution growth method having approximate ...
Microwave-Assisted In Situ Cyclization of Curcumin Derivatives as Dominant Chemotherapeutic Agents for Leukemia and Colon Cancer

Hadiyal, S. D.; Lalpara, J. N.; Dhaduk, B. B. (Pleiades Publishing, Ltd. /Russian Journal of Bioorganic Chemistry, 2022)

A rapid and efficient protocol has been proposed for the synthesis of 7-(4-substituted benzylidene)-3-(4-substituted phenyl)-3,3a,4,5,6,7-hexahydro-2H-indazoles under microwave irradiation. The synthesized compounds were ...
Microwave-Assisted In Situ Cyclization of Curcumin Derivatives as Dominant Chemotherapeutic Agents for Leukemia and Colon Cancer

Hadiyal, S. D.; Lalpara, J. N.; Dhaduk, B. B. (Russian Journal of Organic Chemistry, 2022)

A rapid and efficient protocol has been proposed for the synthesis of 7-(4-substituted benzylidene)-3-(4-substituted phenyl)-3,3a,4,5,6,7-hexahydro-2H-indazoles under microwave irradiation. The synthesized compounds were ...
Microwave-assisted three-component domino synthesis of polysubstituted 4 H-pyran derivatives and their anticancer activity

Hadiyal, S. D.; Parmar, N. D.; Kalavadiya, P. L.; Lalpara, J. N.; Joshi, H. S. (Pleiades Publishing, Ltd. /Russian Journal of Organic Chemistry, 2020)

An efficient microwave-assisted one-pot procedure has been proposed for the synthesis of new4-aryl-6-(methylamino)-5-nitro-2-(1H-pyrrol-2-yl)-4H-pyran-3-carbonitriles by condensation of 3-oxo-3-(1H-pyrrol-2-yl)propanenitrile ...
New 1,3,4-Oxadiazole based Schiff base Derivatives: Synthesis, Characterization and Antibacterial Activity Along With in Silico Studies

Lalpara, J. N.; Hadiyal, S. D.; Dhalani, J. M.; Dubal, G. G. (European chemical bulletin, 2021)

A series of novel 1,3,4-oxadiazole based Schiff base derivatives were designed and synthesized using the efficient strategy with excellent yields. Synthesized molecules evaluated in vitro antibacterial studies in contradiction ...
Palladium‐catalyzed synthesis of novel pyrido [3, 4‐d] pyridazin‐1 (2H)‐ones as promising α‐glucosidase, α‐amylase and EGFR inhibitors along with molecular docking

Radia, A. J.; Lalpara, J. N.; Hadiyal, S. D.; Kaneria, M.; Tirgar, P. R.; Dubal, G. G. (Wiley / Journal of Heterocyclic Chemistry, 2023)

A novel route has been established for the synthesis of novel pyrido[3,4-d]pyri-dazin-1(2H)-one derivative. Synthesis of intermediate 4-methyl-7-(piperazin-1-yl)pyrido[3,4-d]pyridazin-1(2H)-one carried out in the presence ...
Phenylboronic acid catalyzed synthesis of polysubstituted 1,4-dihydropyridine derivatives as promising antioxidant agents correlated with molecular docking

Pansuriya, K.; Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Dubal, G. G (Chemical Data Collections, 2022)

A series of polysubstituted 1, 4-dihydropyridines (4a-i) were designed and developed using Ph-B (OH) 2 catalyst. Further, compounds were confirmed by various spectroscopic techniques. After that all compounds were ...
Rational synthesis, anticancer activity, and molecular docking studies of novel benzofuran liked thiazole hybrids Sanj

Hadiyal, S. D.; Lalpara, J. N.; Dhaduk, B. B.; Joshi, H. S. (Molecular Diversity, 2023)

A novel series of benzofuran bearing thiazole hybrids were synthesized by the multistep reaction approach. All synthesized molecules were selected by the National Cancer Institute, USA for one-dose anticancer activity ...
Synthesis and in vitro antidiabetic screening of novel dihydropyrimidine derivatives

Lalpara, J. N.; Vachhani, M. D.; Hadiyal, S. D.; Goswami, S.; Dubal, G. G. (Pleiades Publishing, Ltd. /Russian Journal of Bioorganic Chemistry, 2021-03-23)

A series of N-substituted-6-methyl-4-{4-[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]methoxyphenyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamides have been synthesized by the condensation of newly synthesized {4-[5-(4-nit ...
Trimethylsilyl chloride catalyzed synthesis of fluoro substituted tetrahydropyrimidines: Molecular docking and antidiabetic studies

Pansuriya, K.; Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Dubal, G. G. (Chemical Data Collections,, 2022)

A novel series of tetrahydropyrimidine derivatives containing azepino indole and aryl substitution was achieved by a multicomponent synthetic approach using Biginelli condensation. Various catalysts were employed in the ...
Water promoted one pot synthesis of sesamol derivatives as potent antioxidants: DFT, molecular docking, SAR and single crystal studies

Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Gupta, M. K.; Solanki, M. B.; Sharon, A.; Dubal, G. G. (Taylor & Francis Group, LLC / Polycyclic Aromatic Compounds, 2022-06-03)

A one pot water mediated synthesis of sesamol analogous using Betti Base synthetic approach. The reaction was optimized with various solvents and catalysts, but the product formed with a high yield in aqueous ethanol ...
Water Promoted One Pot Synthesis of Sesamol Derivatives as Potent Antioxidants: DFT, Molecular Docking, SAR and Single Crystal Studies

Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Gupta, M. K.; Solanki, M. B.; Sharon, A.; Dubal, G. G. (Polycyclic Aromatic Compounds, 2023)

A one pot water mediated synthesis of sesamol analogous using Betti Base synthetic approach. The reaction was optimized with various solvents and catalysts, but the product formed with a high yield in aqueous ethanol ...

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