01. Journal Articles: Recent submissions

Now showing items 41-60 of 154

Stability Indicating RP-UPLC Method for the Quantitative Determination of Degradation Impurities of Benidipine Hydrochloride & Metoprolol Succinate in Combined Dosage Form

Shah, Pranavkumar; Hadiyal, Sanjay; Lalpara, Jaydeep; Dubal, Gaurang; Dhaduk, Bhavin (Springer / Pharmaceutical Chemistry Journal, 2024)

A suitable RP-UPLC method for the quantitative analysis of degradation impurities of Benidipine hydrochloride & Metoprolol succinate is reported. The method was validated for specicity, linearity, range, accuracy, precision, ...
Synthesis of 8-methyl-2-phenylquinazolin-4 (3H)-ones derived Schiff's bases: Spectroscopic properties, SAR, docking approaches and their anticancer and antimicrobial activity

Ramani, Naimish; Patel, Bonny Y.; Italiya, Gopal; Ramalingam, Prasanna Srinivasan; Mishra, Rudra; Subramanian, Sangeetha; Hadiyal, Sanjay D (Elsevier / Journal of Molecular Structure, 2024)

A series of new compounds based on 8-methyl-2-phenyl quinazolinone Schiff's base were synthesized from 3-amino quinazolinone intermediates. These compounds were evaluated for their potential as anticancer and antimicrobial ...
Microwave-Assisted In Situ Cyclization of Curcumin Derivatives as Dominant Chemotherapeutic Agents for Leukemia and Colon Cancer

Hadiyal, S. D.; Lalpara, J. N.; Dhaduk, B. B. (Russian Journal of Organic Chemistry, 2022)

A rapid and efficient protocol has been proposed for the synthesis of 7-(4-substituted benzylidene)-3-(4-substituted phenyl)-3,3a,4,5,6,7-hexahydro-2H-indazoles under microwave irradiation. The synthesized compounds were ...
RP-HPLC In-Vitro Dissolution Method Development and Validation for Determination of Olmesartan Medoxomil, Chlorthalidone and Cilnidipine Drug Combinations

Shah, P.; Dhaduk, B. (2022)

Objective: A simple, sensitive, and accurate in-vitro dissolution method has been developed for Olmesartan Medoxomil (OLM), Chlorthalidone (CHLR) & Cilnidipine (CIL) drug combination according to USP dissolution testing ...
A green one-pot synthetic protocol of hexahydropyrimido [4, 5-d] pyrimidin-4 (1 H)-one derivatives: molecular docking, ADMET, anticancer and antimicrobial studies

Trivedi, Harsh D.; Patel, Bonny Y.; Hadiyal, Sanjay D.; Italiya, Gopal; Ramalingam, Prasanna Srinivasan (Springer Nature Switzerland / Molecular Diversity, 2024)

Ten hexahydropyrimido[4,5-d]pyrimidine derivatives have been synthesized by using a green and time-efficient microwave method. The synthesized motifs were evaluated for their anticancer activity, antimicrobial activity, ...
Water Promoted One Pot Synthesis of Sesamol Derivatives as Potent Antioxidants: DFT, Molecular Docking, SAR and Single Crystal Studies

Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Gupta, M. K.; Solanki, M. B.; Sharon, A.; Dubal, G. G. (Polycyclic Aromatic Compounds, 2023)

A one pot water mediated synthesis of sesamol analogous using Betti Base synthetic approach. The reaction was optimized with various solvents and catalysts, but the product formed with a high yield in aqueous ethanol ...
Stability indicating LC-MS/MS method and validation of selexipag impurities and identification of its force degradation products

Shah, Pranavkumar; Hadiyal, Sanjay D.; Dhaduk, Bhavin B. (Elsevier / Results in Chemistry, 2023-07-05)

Selexipag belongs to a class of medicines known as IP prostacyclin receptor agonists used to treat pulmonary arterial hypertension. A simple and sensitive LC-MS/MS method has been developed for the identification of process ...
Rational synthesis, anticancer activity, and molecular docking studies of novel benzofuran liked thiazole hybrids Sanj

Hadiyal, S. D.; Lalpara, J. N.; Dhaduk, B. B.; Joshi, H. S. (Molecular Diversity, 2023)

A novel series of benzofuran bearing thiazole hybrids were synthesized by the multistep reaction approach. All synthesized molecules were selected by the National Cancer Institute, USA for one-dose anticancer activity ...
Growth and Characterization of Dicoumarole Derivative

Parmar, S. K.; Gohil, H. K.; Vyas, P. M.; Hadiyal, S. D.; Patel, A. H. (International Journal of Advance and Innovative Research, 2018)

The Dicoumarole derivative 4-amino-3-((4-amino-2-oxo-2H-chromen-3-yl)(3-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl)methyl)-2H-chromen-2-one obtain by crystal growth by slow evaporation solution growth method having approximate ...
New 1,3,4-Oxadiazole based Schiff base Derivatives: Synthesis, Characterization and Antibacterial Activity Along With in Silico Studies

Lalpara, J. N.; Hadiyal, S. D.; Dhalani, J. M.; Dubal, G. G. (European chemical bulletin, 2021)

A series of novel 1,3,4-oxadiazole based Schiff base derivatives were designed and synthesized using the efficient strategy with excellent yields. Synthesized molecules evaluated in vitro antibacterial studies in contradiction ...
Trimethylsilyl chloride catalyzed synthesis of fluoro substituted tetrahydropyrimidines: Molecular docking and antidiabetic studies

Pansuriya, K.; Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Dubal, G. G. (Chemical Data Collections,, 2022)

A novel series of tetrahydropyrimidine derivatives containing azepino indole and aryl substitution was achieved by a multicomponent synthetic approach using Biginelli condensation. Various catalysts were employed in the ...
A rapid quantification method for simultaneous determination of pendimethalin and metribuzin contents in suspoemulsion formulation.

Singh, Rakesh; Dhaduk, B.; Dhalani, J. (Results in Chemistry, 2023)

Pendimethalin and metribuzin are combined to a suspoemulsion (SE) formulation that is treated as a pre-emergence and early post emergence herbicide. A simple reverse phase high performance liquid chromatography (RP-HPLC) ...
Rational synthesis, anticancer activity, and molecular docking studies of novel benzofuran liked thiazole hybrids

Hadiyal, Sanjay D.; Lalpara, Jaydeep N.; Dhaduk, Bhavin B.; Joshi, H. S. (Springer Nature Switzerland / Molecular Diversity, 2022-07-19)

A novel series of benzofuran bearing thiazole hybrids were synthesized by the multistep reaction approach. All synthesized molecules were selected by the National Cancer Institute, USA for one-dose anticancer activity ...
Phenylboronic acid catalyzed synthesis of polysubstituted 1, 4-dihydropyridine derivatives as promising antioxidant agents correlated with molecular docking

Pansuriya, Ketan; Lalpara, Jaydeep N.; Hadiyal, Sanjay D.; Dhaduk, Bhavin B.; Dubal, G.G. (Elsevier / Chemical Data Collections, 2022-12)

A series of polysubstituted 1,4-dihydropyridines (4a-i) were designed and developed using Ph-B(OH)2 catalyst. Further, compounds were confirmed by various spectroscopic techniques. After that all compounds were studied for ...
Trimethylsilyl chloride catalyzed synthesis of fluoro substituted tetrahydropyrimidines: Molecular docking and antidiabetic studies

Pansuriya, Ketan; Lalpara, Jaydeep N.; Hadiyal, Sanjay D.; Dhaduk, B.B.; Dubal, G.G. (Elsevier / Chemical Data Collections, 2022-07-14)

A novel series of tetrahydropyrimidine derivatives containing azepino indole and aryl substitution was achieved by a multicomponent synthetic approach using Biginelli condensation. Various catalysts were employed in the ...
Phenylboronic acid catalyzed synthesis of polysubstituted 1,4-dihydropyridine derivatives as promising antioxidant agents correlated with molecular docking

Pansuriya, K.; Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Dubal, G. G (Chemical Data Collections, 2022)

A series of polysubstituted 1, 4-dihydropyridines (4a-i) were designed and developed using Ph-B (OH) 2 catalyst. Further, compounds were confirmed by various spectroscopic techniques. After that all compounds were ...
Biorelevant dissolution studies of platelet aggregation inhibitor: Ticagrelor hydrochloride and its co-crystal with sodium salt of Aspiri

Ambasana, M. A; Kapuriya, N. P.; Ambasana, P. A.; Bhalodia, J.; Bapodra, A. H. (Indian Journal of Chemical Technology, 2022)

The comparative dissolution characteristics of poorly soluble platelet aggregation inhibitor Ticagrelor hydrochloride and its co-crystal with sodium salt of Aspirin in biorelevant media have been demonstrated. The API and ...
Water promoted one pot synthesis of sesamol derivatives as potent antioxidants: DFT, molecular docking, SAR and single crystal studies

Lalpara, J. N.; Hadiyal, S. D.; Dhaduk, B. B.; Gupta, M. K.; Solanki, M. B.; Sharon, A.; Dubal, G. G. (Taylor & Francis Group, LLC / Polycyclic Aromatic Compounds, 2022-06-03)

A one pot water mediated synthesis of sesamol analogous using Betti Base synthetic approach. The reaction was optimized with various solvents and catalysts, but the product formed with a high yield in aqueous ethanol ...
Design and rapid microwave irradiated one-pot synthesis of tetrahydropyrimidine derivatives and their screening in vitro antidiabetic activity

Lalpara, J. N.; Hadiyal, S. D.; Radia, A. J.; Dhalani, J. M.; Dubal, G. G. (Taylor & Francis Group, LLC / Polycyclic Aromatic Compounds, 2020-12-01)

A rapid and efficient method has been developed for one-pot synthesis of some newly designed tetrahydropyrimidine derivatives with aid of 1,3,4-oxadiazole containing aldehyde, substituted acetoacetanilide and thiourea/guanidine ...
Image Set Quality Optimization for Handwritten Gujarati Character and Its Modifier Recognition

Vanjara, Pratik A; Doshi, Priyank D (2022-03-25)

The problem of recognizing handwritten Gujarati characters has been tried by many researchers but still it requires enough work from vowel recognition up to its online application. The problem becomes even more complex if ...

Now showing items 41-60 of 154

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